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森の木

Publications

Please click DOI to access the Web site of original papers.

Original Papers

If you would like to see the original paper, please request it from ResearchGate.

32

One-Pot Conversion of Benzyl Alcohols to N-Protected Anilines and Alkyl Alcohols to Carbamoyl Azides
Kobayashi, S.* Yamaguchi, R.; Yamamoto, F.; Komori, J.; Sakamoto, H. Kasashima, T.; Adriaenssens, L.; Lear, M. J.*
Eur. J. Org. Chem2023, e202300786. DOI: 10.1002/ejoc.202300786

31

Total Synthesis of Geranyl-Resorcinols Isolated from Mushrooms of GenusHericium

Kobayashi, S.;*

Synthesis 202355, 417-432. DOI: 10.1055/a-1944-9623

(This paper was selected for the cover graphic.)

30

Potential Degradation of 4-Methyltetrahydropyran (4-MeTHP) under Oxidation Conditions

Kobayashi, S.;* Tamura, T.

Asian J. Org. Chem. 2021, 10 (10), 2675-2681. DOI: 10.1002/ajoc.202100441

(The art of this paper was selected as a Cover Feature)

29

Cyclopentyl methyl ether (CPME) and 4-methyltetrahydropyran (4-MeTHP): Basic chemical properties and applications as next generation reaction solvents

Kobayashi, S.*

J. Synth. Org. Chem. Jpn 2021 , 79 (6), 547-557. (in Japanese) DOI: 10.5059 / yukigoseikyokaishi.79.547

28

Total Synthesis, Structure Revision and Neuroprotective Effect of Hericenones C–H and Their Derivatives

Kobayashi, S .; * Tamura, T .; Koshishiba, M .; Yasumoto, T .; Shimizu, S .; Kintaka, T .; Nagai, K.

J. Org. Chem. 2021 , 86 (3), 2602-2620. DOI: 10.1021 / acs.joc.0c02681

27

Stereocontrolled Total Synthesis of (+)-Isolaurenidificin and (–)-Bromlaurenidificin

Kobayashi, S .; * Hori, Y .; Yoneyama, R .; Tamura, T .; Masuyama, A.

J. Org. Chem .  2019 , 84 (23), 15549-15556. DOI: 10.1021 / acs.joc.9b02532

26

4-Methyltetrahydropyran (4-MeTHP): Application as an Organic Reaction Solvent

Kobayashi, S .; * Tamura, T .; Yoshimoto, Y .; Kawakami, T .; Masuyama, A.

Chem. Asian J.  2019 , 14 (21), 3921-3937. DOI: 10.1002 / asia.201901169

(This paper was selected for a special collection celebrating 100th Annual Meeting of CSJ)

25

Total syntheses and endoplasmic reticulum stress suppressive activities of hericenes A−C and their derivatives

Kobayashi, S .; * Hamada, Y .; Yasumoto, T .; Hashino, Y .; Masuyama, A .; Nagai, K. *

Tetrahedron Lett .  2018 , 59 (18), 1733-1736. DOI: 10.1016 / j.tetlet.2018.03.065

24

Syntheses of (−)-Tripterifordin and (−)-Neotripterifordin from Stevioside

Kobayashi, S .; * Shibukawa, K .; Hamada, Y .; Kuruma, T .; Kawabata, A .; Masuyama, A.

J. Org. Chem .  2018 , 83 (3), 1606-1613. DOI: 10.1021 / acs.joc.7b02916

23

Grignard Reactions in Cyclopentyl Methyl Ether (CPME)

Kobayashi, S .; * Shibukawa, K .; Miyaguchi, Y .; Masuyama, A.

Asian J. Org. Chem . 2016 , 5 (5), 636-645. DOI: 10.1002 / ajoc.201600059

(Most Accessed 07/2020 to 06/2021) 

22

Stereocontrolled Synthesis of a Possible Stereoisomer of Laurenidificin and a Formal Total Synthesis of (+)-Aplysiallene Featuring a Stereospecific Ring Contraction

Kobayashi, S .; * Yokoi, T .; Inoue, T .; Hori, Y .; Saka, T .; Shimomura, T .; Masuyama, A.

J. Org. Chem . 2016 , 81 (4), 1484-1498. DOI: 10.1021 / acs.joc.5b02595

21

Divergent Total Synthesis of Bioactive Molecules Derived from the Fruiting Bodies of Hericium erinaceum

Kobayashi, S.*

J. Synth. Org. Chem. Jpn 2015 , 73 (2), 131-139. (in Japanese)

DOI: 10.5059 / yukigoseikyokaishi.73.131

20

Divergent Synthesis of Bioactive Resorcinols Isolated from the Fruiting Bodies of Hericium erinaceum: Total Syntheses of Hericenones A, B and I, Hericenols BD, and Erinacerins A and B

Kobayashi, S .; * Tamanoi, H .; Hasegawa, Y .; Segawa, Y .; Masuyama, A.

J. Org. Chem . 2014 , 79 (11), 5227-5238. DOI: 10.1021 / jo500795z

19

Evaluation of Cyclopentyl Methyl Ether (CPME) as a Solvent for Radical Reactions

Kobayashi, S .; * Kuroda, H .; Ohtsuka, Y .; Kashihara, T .; Masuyama, A .; Watanabe, K.

Tetrahedron 2013 , 69 (10), 2251-2259. DOI: 10.1016 / j.tet.2013.01.030

18

Total Synthesis and Structural Revision of Hericerin

Kobayashi, S .; * Inoue, T .; Ando, A .; Tamanoi, H .; Ryu, I .; Masuyama, A.

J. Org. Chem . 2012 , 77 (13), 5819-5822. DOI: 10.1021 / jo300719m

17

Rapid Access to 6-Bromo-5,7-dihydroxyphthalide 5-Methyl Ether by a CuBr2-Mediated Multi-Step Reaction. Concise Total Syntheses of Hericenone J and 5'-Deoxohericenone C (Hericene A)

Kobayashi, S .; * Ando, A .; Kuroda, H .; Ejima, S .; Masuyama, A .; Ryu, I.

Tetrahedron 2011 , 67 (47), 9087-9092. DOI: 10.1016 / j.tet.2011.09.104

16

Stereocontrolled Synthesis of Substituted Bicyclic Ethers through Oxy-Favorskii Rearrangement. Total Synthesis of (±)-Communiol E

Kobayashi, S .; * Kinoshita, T .; Kawamoto, T .; Wada, M .; Kuroda, H .; Masuyama, A .; Ryu, I.

J. Org. Chem . 2011 , 76 (17), 7096-7103. DOI: 10.1021 / jo201064h

(This article was featured in Synfacts 2011 , 11 , 1160.)

15

Black Light Induced Radical Hydroxymethylation of Alkyl Iodides with Atmospheric CO in the Presence of Tetrabutylammonium Borohydride

Kobayashi, S .; Kawamoto, T .; Uehara, S .; Fukuyama, T .; Ryu, I. *

Org. Lett . 2010 , 12 (7), 1548-1551. DOI: 10.1021 / ol1002847

14

Novel Radical Cyclization Method Accompanied by Elimination of Hydrazyl Radical

Kobayashi, S .; Hirao, H .; Kawauchi, T .; Ryu, I. *

Heterocycles 2010 , 80 (2), 879-885. DOI: 10.3987 / COM-09-S (S) 115

13

Organocatalytic Enantioselective Synthesis of Nitrogen-Substituted Dihydropyran-2-one, A Key Synthetic Intermediate of 1β-Methylcarbapenems

Kobayashi, S .; * Uehara, H .; Kinoshita, T .; Sudo, T .; Ryu, I.

Org. Lett . 2009 , 11 (17), 3934-3937. DOI: 10.1021 / ol901544q

12

Enantioselective Synthesis of the Fully Functionalized ABC ring of Zoanthenol

Sugano, N .; Koizumi, Y .; Hirai, G .; Oguri, H .; Kobayashi, S .; Yamashita, S .; Hirama, M. *

Chem. Asian J. 2008 , 3 (8-9), 1549-1557. DOI: 10.1002 / asia.200800079

11

Construction of the CDE-Ring Framework of Erinacine E through Pummerer-type Cyclization

Kobayashi, S .; * Ishii, A .; Toyota, M.

Synlett 2008 , (7), 1086-1090. DOI: 10.1055 / s-2008-1042922

10

Synthesis of trans -Fused Tetrahydrooxepins: Stereoselective Allylation of Sulfur or Fluoro-substituted Tetrahydrooxepins

Kobayashi, S .; * Hori, M .; Hirama, M.

Carbohydr. Res . 2008 , 343 (3), 443-452. DOI: 10.1016 / j.carres. 2007.11.018

09

Radical chain reactions using THP as a solvent

Yasuda, H .; * Uenoyama, Y .; Nobuta, O .; Kobayashi, S .; Ryu, I. *

Tetrahedron Lett . 2008 , 49 (2), 367-370. DOI: 10.1016 / j.tetlet. 2007.11.039

08

Formal Total Synthesis of Neocarzinostatin Chromophore

Kobayashi, S .; * Hori, M .; Wang, GX; Hirama, M. *

J. Org. Chem . 2006 , 71 (2), 636-644. DOI: 10.1021 / jo052031o

07

Stereocontrolled Synthesis of the ABCDE Ring Moiety of Ciguatoxin CTX3C

Kobayashi, S .; Takahashi, Y .; Komano, K .; Alizadeh, BH, Kawada, Y .; Oishi, T .; Tanaka, S .; Ogasawara, Y .; Sasaki, S .; Hirama, M. *

Tetrahedron 2004 , 60 (38), 8375-8396. DOI: 10.1016 / j.tet.2004.07.010

06

Total Synthesisof 9-Membered Enediyne Antibiotic N1999-A2: Absolute Stereochemistry and DNA Cleavage

Kobayashi, S.; * Hirama, M. *

J. Synth. Org. Chem. Jpn 2004 , 62 (3), 184-193. (in Japanese)

DOI: 10.5059 / yukigoseikyokaishi.62.184

05

Synthesis of the Fully Functionalized ABCDE Ring Moiety of Ciguatoxin

Kobayashi, S .; Alizadeh, BH; Sasaki, S .; Oguri, H .; Hirama, M. *

Org. Lett. 2004 , 6 (5), 751-754. DOI: 10.1021 / ol0364475

04

Diastereoselective Additions of Ethynyl Grignard Reagent to Erythrulose Derivatives

Kobayashi, S .; Das, P .; Wang, GX; Mita, T .; Lear, MJ; Hirama, M. *

Chem. Lett . 2002 , (3), 300-301. DOI: 10.1246 / cl.2002.300

03

The First Total Synthesis of N1999-A2: Absolute Stereochemistry and Stereochemical Implications into DNA Cleavage

Kobayashi, S .; Ashizawa, S .; Takahashi, Y .; Sugiura, Y .; Nagaoka, M .; Lear, MJ; Hirama, M. *

J. Am Chem. Soc . 2001 , 123 (45), 11294-11295. DOI: 10.1021 / ja003982g

02

Investigation of the Total Synthesis of N1999-A2: Implication of Stereochemistry

Kobayashi, S .; Reddy, RS; Sugiura, Y .; Sasaki, D .; Miyagawa, N .; Hirama, M. *

J. Am Chem. Soc . 2001 , 123 (12), 2887-2888. DOI: 10.1021 / ja011779v

01

Palladium-Catalyzed Coupling of Alkenyl Iodides with Ethynyl Oxiranes: Synthesis of Epoxy Enediyne Core Intermediates Related to Neocarzinostatin Chromophore

Reddy, RS; Iguchi, S .; Kobayashi, S .; Hirama, M. *

Tetrahedron Lett . 1996 , 37 (52), 9335-9336. DOI: 10.1016 / S0040-4039 (97) 82957-7

Original Papers
Others
Others

03

Stereocontrolled total synthesis and structure determination of brominated natural products isolated from red algae

Kobayashi, S.*

AgriBio 2024, 8 (9), 752-754. ISBN: 01327-08

02

Development of suppressive agents against endoplasmic reticulum stress-dependent neuronal cell death

Kobayashi, S.*

The Cell 2022, 54 (4), 226-228. ISBN: 17601-04

01

Development of neuroprotective agents effective for prevention and improvement of cognitive disorder

Kobayashi, S.*

AgriBio 2021, 5 (12), 1055-1058. ISBN: 01327-11

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